Clomiphene Citrate – a popular anti-estrogenic drug Greek production, which is based on the eponymous substance clomiphene. By the properties of this estrogen receptor blocker. In sports, it applies no less than in medical practice. In sports practice for its reception resort athletes who use anabolic and androgenic steroids – to restore natural levels of testosterone and estrogen to prevent side effects.
In medicine Clomiphene citrate is prescribed mainly for ovarian stimulation and therapy / treatment of disorders that prevent conception. Indications are as follows: when androgen deficiency, with polycystic ovaries, with anovulatory infertility, with oligospermia and other prescription.
Description Clomiphene Citrate
As mentioned, the active ingredient of this drug is the same name his substance. Clomiphene – is in high demand antagonist of estrogen in their chemical structure most similar to tamoxifen. Demand for it provided useful properties, which, although they are not very multiplicity, but handy for the treatment of humans, and to support athletes who use anabolic and androgenic steroids for the purpose of improvement of physical fitness.
The most valuable for athletes are the following properties of clomiphene citrate
• First, its ability to increase the production of testosterone (effect on the HPTA axis (hypothalamic – pituitary – testes and increases the synthesis of LH and follicle-stimulating hormone, which in turn increases and production of natural testosterone);
• Second, its antiestrogenic quality (blocking estradiol and estrogen receptors in cells with estrogen production process itself, aromatization is not blocked or slowed expressed).
On the practical side, all these effects and actions exhibited by Clomiphene citrate, are primarily aimed at protecting the athlete from disorders associated with taking steroids. More specifically, this drug vo-pervyh, provides protection from the adverse effects of estrogen (gynecomastia, increased fat and OE), and vo-vtoryh, protects against the loss of muscle mass gained during the course (normalizes the production of testosterone, the thus prevents the strengthening of catabolic processes).
It is also known that applying in accordance with the recommendations tablets Clomiphene Citrate production contribute to the prevention of osteoporosis (due to the activation of estrogen receptors, which are located in the bone).
Note that no self Clomiphene Citrate shows no side effects, that is, it is practically not inherent side effects.In fact, any deviations from the norm can be observed only in overdose, especially in the use of very high doses may disturb you dizziness, headaches, nausea, blurred vision (passing a character).
In conclusion, the storage of tablets of the drug, it is desirable to carry out protected from light and moisture.Storage temperature should not exceed the room rate. Keep away from children and pets.
How to receive clomiphene citrate?
To begin with: to use the anti-estrogen is recommended for sport exclusively for men. And all because women athletes by implementing long-term use of these tablets may be faced with a violation of the natural level of hormones in the body. The most terrible thing that can happen to an athlete – a nausea, headaches, blurred vision and dizziness in overdose. So the men in sport who use pills of clomiphene, and listen to the recommendations, there is practically nothing to fear.
It is important that the use of clomiphene citrate is recommended to start almost immediately after the completion of steroids, literally the next day. So, you will ensure maximum security yourself from the “rollback phenomenon” and the subsequent loss of muscle mass gained during the course.
What else you need to know the athlete planner FCT with the drug? Firstly, the average dosage of clomiphene citrate is 50-150 mg per day. Secondly, it is desirable to use the pill daily, at one and the same time, drinking plenty of fluids (avoid alcohol intake). Third, that the use of the drug takes an average of two to three full weeks.And fourthly, that the dosage and duration vary considerably depending on the current course.
Specify that calculate the dose that you know you need it the dose, simply because it has a convenient concentration of the active substance – 50 mg / tab. And indeed, it is practically impossible to make a mistake, because it turns out that for the reception of the most-recommended dose (150 mg) should be exactly 3 tablets of the drug for an average dose (100 mg) – 2 tablets, and for the minimum recommended (50 mg) – one.
Note: for more information on how to take Clomiphene Citrate, visit our forum. Here you can chat with experienced consultants (masters of different sports, sports physician, and others.) And get useful tips on the best practice.
Reviews of Clomiphene Citrate
To learn about the qualities of this drug other people think athletes do not need long to “wander” through the network. Just go to our forum and study there feedback left by customers. We have never restricted the visitors desire to communicate, so on our website is not observed a lack of relevant, useful and important information for the study of what is called a “first-hand”.
Visit the forums and reading reviews about Clomiphene Citrate, you make sure that the anti-estrogenic drug comes in handy not only to counter the effects of the reception aromatizing steroid (gynecomastia, fluid retention, increase in body fat), but also to prevent the so hated athletes “rollback phenomenon”. For reference: the “rollback phenomenon” – is the process of reduction of muscle mass caused by insufficient production of testosterone.
As the anti-estrogen is struggling with it? It’s simple: as the guide suggests, the active substance affects the HPTA axis, increasing the synthesis of gonadotropins, which are involved in the production of natural testosterone.
However, this drug like athletes not only for their effectiveness. There he and other equally nice quality, such as practicality. What is it? A convenient concentration of the active substance, which is prompt feedback makes it easy to calculate the dose needed to. Make a mistake here will be difficult.
It is important that Clomiphene Citrate boasts of its safety for humans. He hardly peculiar side effects, and those that may arise, often manifested in overdose (headaches, visual haze, nausea). So the athlete to listen to the recommendations to be afraid of almost nothing.
Clomiphene Citrate is typically prescribed for women to aid in ovulation. In men, the application of Clomid causes an elevation of follicle stimulating hormone and luteinizing hormone. As a result, natural testosterone production is also increased.
This effect is obviously beneficial to the athlete, especially at the conclusion of a steroid cycle when endogenous testosterone levels are subnormal. When an athlete discontinues the use of steroids, his testosterone levels will most likely be suppressed. If endogenous testosterone levels are not brought to normal, a dramatic loss in size and strength may occur. Clomid plays a crucial role in preventing this crash in athletic performance.
Bodybuilders find that a daily intake of 50-100 mg of clomiphene citrate over a two week period will bring endogenous testosterone production back to an acceptable level. Clomid will gradually raise testosterone levels over its period of intake. Since an immediate boost in testosterone is often desirable, athlete will commonly use HCG (human choronic gonadotropin) for a couple of weeks, and the continue treatment with Clomid.
Clomid is also effective as an anti-estrogen. Most athletes will suffer from an elevated estrogen level at the conclusion of a cycle. A high estrogen level combined with a low testosterone level puts an athlete in serious risk of developing gynocomastia. With the intake of Clomid, the athlete gets the dual effect of blocking out some of the effects of estrogen, while also increasing endogenous testosterone production.